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BIX 01294 Trihydrochloride
CAS No. 1392399-03-9
BIX 01294 Trihydrochloride ( —— )
Catalog No. M11632 CAS No. 1392399-03-9
BIX01294 is an inhibitor of G9a histone methyltransferase with IC50 of 2.7 μM in a cell-free assay.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 45 | In Stock |
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| 5MG | 59 | In Stock |
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| 10MG | 98 | In Stock |
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| 25MG | 182 | In Stock |
|
| 50MG | 259 | In Stock |
|
| 100MG | 466 | In Stock |
|
| 500MG | 1044 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBIX 01294 Trihydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionBIX01294 is an inhibitor of G9a histone methyltransferase with IC50 of 2.7 μM in a cell-free assay.
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DescriptionBIX01294 is an inhibitor of G9a histone methyltransferase with IC50 of 2.7 μM in a cell-free assay, reduces H3K9me2 of bulk histones, also weakly inhibits GLP (primarily H3K9me3), no significant activity observed at other histone methyltransferases.
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetHMTase
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RecptorG9a
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Research AreaOther Indications
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Indication——
Chemical Information
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CAS Number1392399-03-9
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Formula Weight600.02
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Molecular FormulaC28H38N6O2·3HCl
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Purity>98%(HPLC)
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SolubilityEthanol: 8 mg/mL (13.33 mM); Water: 98 mg/mL (163.32 mM); DMSO: 98 mg/mL (163.32 mM)
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SMILESCl.Cl.Cl.COC1=C(OC)C=C2C(NC3CCN(CC4=CC=CC=C4)CC3)=NC(=NC2=C1)N1CCCN(C)CC1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Kubicek S, et al. Mol Cell, 2007, 25(3), 473-48
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